Entomotherapy is the use of insects and their products for medicinal purposes. Since ancient times, humans have been utilizing insects and their products as a source of medicine for curing ailments due to their antirheumatic, anticancer, immunological, diuretic, analgesic, antibacterial, and anesthetic properties. Insects have long been used in traditional medicine for their useful natural products such as propolis, pollen, bee wax, and royal jelly. The intriguing ways that insects and their products are transforming healthcare are examined in this article.